SKU: T70403-25mg-TM
VUF14480
Blue Ice
Specifications
| Specification | Details |
|---|---|
| Additional Information | VUF14480 is a covalent partial agonist that interacts with cysteine 98(3.36) of the human histamine H₄ receptor. VUF14480 was shown to be a partial agonist of hH4 receptor-mediated G protein signalling and β-arrestin2 recruitment. VUF14480 bound covalently to the hH₄ receptor with submicromolar affinity. Serine substitution of C98(3.36) prevented this covalent interaction. |
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Datasheet
Catalog Number
T70403-25mg-TM
Name
VUF14480
Price(25 mg)
Pack Size