SKU: T21548-10mg-TM
PF-4981517
Blue Ice
Specifications
| Specification | Details |
|---|---|
| Additional Information | PF-4981517 (CYP3cide) is a efficient, specific and time-dependent inhibitor of cytochrome P4503A4 (CYP3A4). The IC 50 values for CYP3A activity are 0.03 μM,17 μM, and 71 μM for CYP3A4, CYP3A5, and CYP3A7, respectively. PF-4981517 is able to be used to distinguish the contributions of CYP3A4 versus CYP3A5 on drug Metabolism. |
| Synonyms | CYP3cide |
Resources
PDF
Datasheet
Catalog Number
T21548-10mg-TM
Name
PF-4981517
Price(10 mg)
Pack Size