SKU: T9564-50mg-TM
IRE1α kinase-IN-1
Blue Ice
Specifications
| Specification | Details |
|---|---|
| Additional Information | IRE1α kinase-IN-1 is a highly selective IRE1α (ERN1) inhibitor, with an IC50 of 77 nM. It displays 100-fold selectivity for IRE1α over the IRE1β isoform. It inhibits ER stress-induced IRE1α oligomerization and autophosphorylation, and also inhibits IRE1α RNase activity (IC50=80 nM) |
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Catalog Number
T9564-50mg-TM
Name
IRE1alpha kinase-IN-1
Price(50 mg)
Pack Size